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GENERAL
TITLE
DOUBLING THE SIZE OF THE GLUCOCORTICOID RECEPTOR LIGAND BINDING POCKET BY DEACYLCORTIVAZOL
DATE LAST MODIFIED
20 Oct 2021
RELEASE
15 Jan 2008
OBSOLETE
CLASSIFICATION
PROTEIN BINDING
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 62
RESOLUTION RANGE HIGH
2.5
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1128/MCB.01541-07
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P04150 NR3C1, GRL ESCHERICHIA COLI BL21(DE3) HUMAN
GR, NUCLEAR RECEPTOR SUBFAMILY 3 GROUP C MEMBER 1
Mutations
Q56404 -- -- --
NCOA-1, STEROID RECEPTOR COACTIVATOR 1, SRC-1, RIP ...
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402