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GENERAL
TITLE
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRDT IN COMPLEX WITH THE INHIBITOR JQ1
DATE LAST MODIFIED
29 Aug 2012
RELEASE
11 Jul 2012
OBSOLETE
CLASSIFICATION
TRANSCRIPTION REGULATOR/INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 2 21
RESOLUTION RANGE HIGH
2.2
RESOLUTION RANGE LOW
42.84
PUBMED ID
DOI
10.1016/J.CELL.2012.06.045
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P00447 BRDT ESCHERICHIA COLI HUMAN
CANCER/TESTIS ANTIGEN 9, CT9, RING3-LIKE PROTEIN
Q13526 BRDT ESCHERICHIA COLI HUMAN
CANCER/TESTIS ANTIGEN 9, CT9, RING3-LIKE PROTEIN
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402