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GENERAL
TITLE
STRUCTURE OF HS/ACPRC2 IN COMPLEX WITH 5,8-DICHLORO-2-[(4-METHOXY-6- METHYL-2-OXO-1,2-DIHYDROPYRIDIN-3-YL)METHYL]-7-[(R)-METHOXY(OXETAN-3- YL)METHYL]-3,4-DIHYDROISOQUINOLIN-1(2H)-ONE
DATE LAST MODIFIED
21 Feb 2018
RELEASE
27 Dec 2017
OBSOLETE
CLASSIFICATION
TRANSFERASE/TRANSFERASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1 21 1
RESOLUTION RANGE HIGH
2.81
RESOLUTION RANGE LOW
148.01
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.7B01375
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P02766 | EZH2 | SPODOPTERA FRUGIPERDA | GREEN ANOLE | -- | ||
Q0TTB4 | EZH2 | SPODOPTERA FRUGIPERDA | GREEN ANOLE | -- | ||
P02741 | EED | SPODOPTERA FRUGIPERDA | HUMAN | HEED,EMBRYONIC ECTODERM DEVELOPMENT PROTEIN,WD PRO ... | ||
P02741 | EED | SPODOPTERA FRUGIPERDA | HUMAN | HEED,EMBRYONIC ECTODERM DEVELOPMENT PROTEIN,WD PRO ... | ||
Q0TTB4 | SUZ12, CHET9, JJAZ1, KIAA0160 | SPODOPTERA FRUGIPERDA | HUMAN | CHROMATIN PRECIPITATED E2F TARGET 9 PROTEIN,CHET 9 ... | ||
P02741 | SUZ12, CHET9, JJAZ1, KIAA0160 | SPODOPTERA FRUGIPERDA | HUMAN | CHROMATIN PRECIPITATED E2F TARGET 9 PROTEIN,CHET 9 ... |
NGL Viewer is used for the molecular visualization.
- AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
- AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402