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GENERAL
TITLE
FRAGMENT-BASED DISCOVERY OF POTENT AND SELECTIVE DDR1/2 INHIBITORS
DATE LAST MODIFIED
-
RELEASE
5 Aug 2015
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
1.9
RESOLUTION RANGE LOW
33
PUBMED ID
DOI
10.1021/ACSMEDCHEMLETT.5B00143

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q08345 DDR1, CAK, EDDR1, NEP, NTRK4, PTK3A, RTK6, TRKE SPODOPTERA FRUGIPERDA HUMAN
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1,CD167 ANTIG ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402