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GENERAL
TITLE
CREBBP BROMODOMAIN IN COMPLEX WITH CPD 44 (3-((5-ACETYL-1- (CYCLOPROPYLMETHYL)-4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[4,3-C]PYRIDIN-3- YL)AMINO)-N-ISOPROPYLBENZAMIDE)
DATE LAST MODIFIED
21 Dec 2016
RELEASE
2 Nov 2016
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1 21 1
RESOLUTION RANGE HIGH
1.087
RESOLUTION RANGE LOW
44.395
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.6B01022
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P28066 CREBBP, CBP ESCHERICHIA COLI HUMAN --
P62191 CREBBP, CBP ESCHERICHIA COLI HUMAN --
P28066 CREBBP, CBP ESCHERICHIA COLI HUMAN --
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402