5M96 logo

5M96

3D Structure View

Loading...

More Info

GENERAL
TITLE
SYNTHESIS AND BIOLOGICAL EVALUATION OF NEW TRIAZOLO AND IMIDAZOLOPYRIDINE RORGT INVERSE AGONISTS
DATE LAST MODIFIED
19 Dec 2018
RELEASE
14 Dec 2016
OBSOLETE
CLASSIFICATION
TRANSCRIPTION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 61
RESOLUTION RANGE HIGH
1.77
RESOLUTION RANGE LOW
19.87
PUBMED ID
DOI
10.1002/CMDC.201600500
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P51449 RORC, NR1F3, RORG, RZRG ESCHERICHIA COLI BL21 HUMAN
NUCLEAR RECEPTOR RZR-GAMMA,NUCLEAR RECEPTOR SUBFAM ...
Mutations
P51449 RORC, NR1F3, RORG, RZRG ESCHERICHIA COLI BL21 HUMAN
NUCLEAR RECEPTOR RZR-GAMMA,NUCLEAR RECEPTOR SUBFAM ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402