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GENERAL
TITLE
BROMODOMAIN OF HUMAN GCN5 WITH 4-BROMO-2-METHYL-5-(((3R,5R)-1-METHYL- 5-PHENYLPIPERIDIN-3-YL)AMINO)PYRIDAZIN-3(2H)-ONE
DATE LAST MODIFIED
24 Jan 2018
RELEASE
20 Dec 2017
OBSOLETE
CLASSIFICATION
TRANSCRIPTION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
1.8
RESOLUTION RANGE LOW
38.84
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.6B01566
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P03372 KAT2A, GCN5, GCN5L2, HGCN5 ESCHERICHIA COLI HUMAN
GENERAL CONTROL OF AMINO ACID SYNTHESIS PROTEIN 5- ...
Q15596 KAT2A, GCN5, GCN5L2, HGCN5 ESCHERICHIA COLI HUMAN
GENERAL CONTROL OF AMINO ACID SYNTHESIS PROTEIN 5- ...
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402