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GENERAL
TITLE
INDOLE-2 CARBOXAMIDES AS SELECTIVE SECRETED PHOSPHOLIPASE A2 TYPE X (SPLA2-X) INHIBITORS
DATE LAST MODIFIED
5 May 2021
RELEASE
1 Aug 2018
OBSOLETE
CLASSIFICATION
LIPID BINDING PROTEIN
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
1.9
RESOLUTION RANGE LOW
44.083
PUBMED ID
DOI
10.1021/ACSMEDCHEMLETT.7B00505
PDBe
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Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonyms | Actions | ||
---|---|---|---|---|---|---|---|---|
O15496 | PLA2G10 | ESCHERICHIA COLI BL21(DE3) | HUMAN | GROUP X SECRETORY PHOSPHOLIPASE A2,SPLA2-X,PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE 10 | HUMAN | GROUP X SECRETORY PHOSPHOLIPASE A2,SPLA2-X,PHOSPHA ... | Mutations | |
O15496 | PLA2G10 | ESCHERICHIA COLI BL21(DE3) | HUMAN | GROUP X SECRETORY PHOSPHOLIPASE A2,SPLA2-X,PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE 10 | HUMAN | GROUP X SECRETORY PHOSPHOLIPASE A2,SPLA2-X,PHOSPHA ... | Mutations |
NGL Viewer is used for the molecular visualization.
- AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
- AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402