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GENERAL
TITLE
CRYSTAL STRUCTURE OF HUMAN MDM2 IN COMPLEX WITH A 12-MER LYSINE- CYSTEINE SIDE CHAIN DITHIOCARBAMATE STAPLED PEPTIDE INHIBITOR PMI
DATE LAST MODIFIED
11 Dec 2019
RELEASE
25 Apr 2018
OBSOLETE
CLASSIFICATION
LIGASE/LIGASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 2 2 21
RESOLUTION RANGE HIGH
1.8
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1039/C8SC03275K
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P52565 | -- | -- | HUMAN | DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ... | ||
P22629 | -- | -- | SYNTHETIC CONSTRUCT | -- | ||
Q00987 | -- | -- | HUMAN | DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ... | Mutations | |
-- | -- | SYNTHETIC CONSTRUCT | -- | |||
P0CG64 | -- | -- | HUMAN | DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ... | ||
-- | -- | SYNTHETIC CONSTRUCT | -- | |||
Q00987 | -- | -- | HUMAN | DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ... | Mutations | |
-- | -- | SYNTHETIC CONSTRUCT | -- | |||
Q00987 | -- | -- | HUMAN | DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ... | Mutations | |
-- | -- | SYNTHETIC CONSTRUCT | -- |