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GENERAL
TITLE
CRYSTAL STRUCTURE OF HUMAN MDM2 IN COMPLEX WITH A 12-MER LYSINE- CYSTEINE SIDE CHAIN DITHIOCARBAMATE STAPLED PEPTIDE INHIBITOR PMI
DATE LAST MODIFIED
11 Dec 2019
RELEASE
25 Apr 2018
OBSOLETE
CLASSIFICATION
LIGASE/LIGASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 2 2 21
RESOLUTION RANGE HIGH
1.8
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1039/C8SC03275K
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P19803 -- -- HUMAN
DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ...
P22629 -- -- SYNTHETIC CONSTRUCT --
Q00987 -- -- HUMAN
DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ...
Mutations
-- -- SYNTHETIC CONSTRUCT --
P0CG64 -- -- HUMAN
DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ...
-- -- SYNTHETIC CONSTRUCT --
Q00987 -- -- HUMAN
DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ...
Mutations
-- -- SYNTHETIC CONSTRUCT --
Q00987 -- -- HUMAN
DOUBLE MINUTE 2 PROTEIN,HDM2,ONCOPROTEIN MDM2,RING ...
Mutations
-- -- SYNTHETIC CONSTRUCT --
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402