5WMD logo

5WMD

3D Structure View

Loading...

More Info

GENERAL
TITLE
N-TERMINAL BROMODOMAIN OF BRD4 IN COMPLEX WITH OTX-015
DATE LAST MODIFIED
13 Feb 2019
RELEASE
1 Aug 2018
OBSOLETE
CLASSIFICATION
TRANSCRIPTION/TRANSCRIPTION INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
1.18
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1158/2159-8290.CD-17-0902
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
O60885 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402