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GENERAL
TITLE
NOVEL BINDING MODES OF INHIBITION OF WILD-TYPE IDH1: ALLOSTERIC INHIBITION WITH CMPD2
DATE LAST MODIFIED
22 Aug 2018
RELEASE
25 Jul 2018
OBSOLETE
CLASSIFICATION
OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 1 2 1
RESOLUTION RANGE HIGH
2.17
RESOLUTION RANGE LOW
137.44
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.8B00305
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P04275 | IDH1, PICD | ESCHERICHIA COLI | HUMAN | IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ... | ||
Q9UIF8 | IDH1, PICD | ESCHERICHIA COLI | HUMAN | IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ... | ||
P72065 | IDH1, PICD | ESCHERICHIA COLI | HUMAN | IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ... | ||
P07359 | IDH1, PICD | ESCHERICHIA COLI | HUMAN | IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ... | ||
P72065 | IDH1, PICD | ESCHERICHIA COLI | HUMAN | IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ... | ||
P0A1I9 | IDH1, PICD | ESCHERICHIA COLI | HUMAN | IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ... |