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GENERAL
TITLE
NOVEL BINDING MODES OF INHIBITION OF WILD-TYPE IDH1: ALLOSTERIC INHIBITION WITH CMPD2
DATE LAST MODIFIED
22 Aug 2018
RELEASE
25 Jul 2018
OBSOLETE
CLASSIFICATION
OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 1 2 1
RESOLUTION RANGE HIGH
2.17
RESOLUTION RANGE LOW
137.44
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.8B00305

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P04275 IDH1, PICD ESCHERICHIA COLI HUMAN
IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ...
Q9UIF8 IDH1, PICD ESCHERICHIA COLI HUMAN
IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ...
P72065 IDH1, PICD ESCHERICHIA COLI HUMAN
IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ...
P07359 IDH1, PICD ESCHERICHIA COLI HUMAN
IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ...
P72065 IDH1, PICD ESCHERICHIA COLI HUMAN
IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ...
P0A1I9 IDH1, PICD ESCHERICHIA COLI HUMAN
IDH,CYTOSOLIC NADP-ISOCITRATE DEHYDROGENASE,IDP,NA ...
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402