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GENERAL
TITLE
STRUCTURE OF PRMT5:MEP50 IN COMPLEX WITH LLY-283, A POTENT AND SELECTIVE INHIBITOR OF PRMT5, WITH ANTITUMOR ACTIVITY
DATE LAST MODIFIED
8 Aug 2018
RELEASE
16 May 2018
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
I 2 2 2
RESOLUTION RANGE HIGH
2.8
RESOLUTION RANGE LOW
61
PUBMED ID
DOI
10.1021/ACSMEDCHEMLETT.8B00014
PDBe
LIGANDS
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P32379 | PRMT5, HRMT1L5, IBP72, JBP1, SKB1 | SPODOPTERA FRUGIPERDA | HUMAN | 72 KDA ICLN-BINDING PROTEIN,HISTONE-ARGININE N-MET ... | ||
P32379 | WDR77, MEP50, WD45, HKMT1069, NBLA10071 | SPODOPTERA FRUGIPERDA | HUMAN | MEP-50,ANDROGEN RECEPTOR COFACTOR P44,WD REPEAT-CO ... |