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GENERAL
TITLE
STRUCTURE OF CDK12/CYCK IN COMPLEX WITH A SMALL MOLECULE INHIBITOR N- (4-(1-METHYL-1H-PYRAZOL-4-YL)PHENYL)-N-((1R,4R)-4-(QUINAZOLIN-2- YLAMINO)CYCLOHEXYL)ACETAMIDE
DATE LAST MODIFIED
26 Sept 2018
RELEASE
29 Aug 2018
OBSOLETE
CLASSIFICATION
TRANSFERASE/INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
2.75
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.8B00683
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
O75909 | CDK12, CRK7, CRKRS, KIAA0904 | UNIDENTIFIED BACULOVIRUS | HUMAN | CDC2-RELATED KINASE,ARGININE/SERINE-RICH,CRKRS,CEL ... | ||
Q9RF12 | CCNK, CPR4 | UNIDENTIFIED BACULOVIRUS | HUMAN | -- | ||
O75909 | CDK12, CRK7, CRKRS, KIAA0904 | UNIDENTIFIED BACULOVIRUS | HUMAN | CDC2-RELATED KINASE,ARGININE/SERINE-RICH,CRKRS,CEL ... | ||
Q9RF12 | CCNK, CPR4 | UNIDENTIFIED BACULOVIRUS | HUMAN | -- |