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GENERAL
TITLE
UNDERSTANDING THE SPECIES SELECTIVITY OF MYELOID CELL LEUKEMIA-1 (MCL- 1) INHIBITORS
DATE LAST MODIFIED
29 Jul 2020
RELEASE
1 Aug 2018
OBSOLETE
CLASSIFICATION
SIGNALING PROTEIN/INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1
RESOLUTION RANGE HIGH
2.7
RESOLUTION RANGE LOW
30
PUBMED ID
DOI
10.1021/ACS.BIOCHEM.8B00626
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P42574 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
P97287 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
Mutations
Q9H2K2 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
Q9H2K2 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
P97287 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
Mutations
P97287 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
Mutations
Q9H2K2 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
P97287 MALE, B4034, JW3994, MCL1 ESCHERICHIA COLI MOUSE
MBP,MMBP,MALTODEXTRIN-BINDING PROTEIN,BCL-2-RELATE ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402