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GENERAL
TITLE
N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH : 8-(((1R,2R,3R,5S)-2-(2-(4, 4-DIFLUOROCYCLOHEXYL)ETHYL)-8-AZABICYCLO[3.2.1]OCTAN-3-YL)AMINO)-3- METHYL-5-(5-METHYLPYRIDIN-3-YL)-1,7-NAPHTHYRIDIN-2(1H)-ONE
DATE LAST MODIFIED
10 Oct 2018
RELEASE
26 Sept 2018
OBSOLETE
CLASSIFICATION
TRANSCRIPTION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 2
RESOLUTION RANGE HIGH
1.7
RESOLUTION RANGE LOW
29.37
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.8B00862
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
Q13563 | BRD4, HUNK1 | ESCHERICHIA COLI | HUMAN | PROTEIN HUNK1 |