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GENERAL
TITLE
CRYSTAL STRUCTURE OF MRIPK3 COMPLEXED WITH N-(3-FLUORO-4-{1H- PYRROLO[2,3-B]PYRIDIN-4-YLOXY}PHENYL)-1-(4-FLUOROPHENYL)-2-OXO-1,2- DIHYDROPYRIDINE-3-CARBOXAMIDE
DATE LAST MODIFIED
1 Apr 2020
RELEASE
17 Jul 2019
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 1 2 1
RESOLUTION RANGE HIGH
2.1
RESOLUTION RANGE LOW
47.53
PUBMED ID
DOI
10.1021/ACSMEDCHEMLETT.9B00065
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q9QZL0 RIPK3, RIP3 SPODOPTERA FRUGIPERDA MOUSE
RIP-LIKE PROTEIN KINASE 3, RECEPTOR-INTERACTING PR ...
Mutations
Q9QZL0 RIPK3, RIP3 SPODOPTERA FRUGIPERDA MOUSE
RIP-LIKE PROTEIN KINASE 3, RECEPTOR-INTERACTING PR ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402