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GENERAL
TITLE
CRYSTAL STRUCTURE OF HUMAN KRAS G12C COVALENTLY BOUND TO AN ACRYLOYLAZETIDINE ACETAMIDE INHIBITOR.
DATE LAST MODIFIED
2 Oct 2019
RELEASE
28 Aug 2019
OBSOLETE
CLASSIFICATION
SIGNALING PROTEIN/INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1
RESOLUTION RANGE HIGH
2.1
RESOLUTION RANGE LOW
30
PUBMED ID
DOI
10.1021/ACSMEDCHEMLETT.9B00258
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P0A3M6 | KRAS, KRAS2, RASK2 | ESCHERICHIA COLI BL21(DE3) | HUMAN | K-RAS 2,KI-RAS,C-K-RAS,C-KI-RAS | ||
O94925 | KRAS, KRAS2, RASK2 | ESCHERICHIA COLI BL21(DE3) | HUMAN | K-RAS 2,KI-RAS,C-K-RAS,C-KI-RAS | ||
P37798 | KRAS, KRAS2, RASK2 | ESCHERICHIA COLI BL21(DE3) | HUMAN | K-RAS 2,KI-RAS,C-K-RAS,C-KI-RAS | ||
O94925 | KRAS, KRAS2, RASK2 | ESCHERICHIA COLI BL21(DE3) | HUMAN | K-RAS 2,KI-RAS,C-K-RAS,C-KI-RAS |