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GENERAL
TITLE
BRD4_BROMODOMAIN2 COMPLEX WITH PYRROLOPYRIDONE COMPOUND 18
DATE LAST MODIFIED
10 Jun 2020
RELEASE
6 May 2020
OBSOLETE
CLASSIFICATION
SIGNALING PROTEIN
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 1 2 1
RESOLUTION RANGE HIGH
2.116
RESOLUTION RANGE LOW
82.94
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.0C00628
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
O60885 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
Mutations
Q14186 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
Q4L5E3 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
Q4L5E4 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402