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GENERAL
TITLE
DISCOVERY OF SARXXXX92, A PAN-PIM KINASE INHIBITOR, EFFICACIOUS IN A KG1 TUMOR MODEL
DATE LAST MODIFIED
25 Nov 2020
RELEASE
4 Nov 2020
OBSOLETE
CLASSIFICATION
ONCOPROTEIN,TRANSFERASE/INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 65
RESOLUTION RANGE HIGH
1.74
RESOLUTION RANGE LOW
86
PUBMED ID
DOI
10.1016/J.BMCL.2020.127625
PDBe
LIGANDS
628 ,
NGL Viewer is used for the molecular visualization.
- AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
- AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402