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GENERAL
TITLE
X-RAY CRYSTAL STRUCTURE OF DASATINIB (BMS-354825) BOUND TO ACTIVATED ABL KINASE DOMAIN
DATE LAST MODIFIED
18 Oct 2017
RELEASE
21 Nov 2006
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 43 21 2
RESOLUTION RANGE HIGH
2.4
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1158/0008-5472.CAN-05-4187
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P00519 | ABL1, ABL, JTK7 | SPODOPTERA FRUGIPERDA | HUMAN | P150, C- ABL, ABELSON MURINE LEUKEMIA VIRAL ONCOGE ... | Mutations | |
P00519 | ABL1, ABL, JTK7 | SPODOPTERA FRUGIPERDA | HUMAN | P150, C- ABL, ABELSON MURINE LEUKEMIA VIRAL ONCOGE ... | Mutations |