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GENERAL
TITLE
DISCOVERY AND OPTIMIZATION OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS FOR THE TREATMENT OF PHOSPHATASE AND TENSIN HOMOLOGUE (PTEN)-DEFICIENT CANCERS
DATE LAST MODIFIED
8 May 2019
RELEASE
15 Jan 2014
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
2.8
RESOLUTION RANGE LOW
154.9
PUBMED ID
DOI
10.1021/JM401642Q
PDBe
LIGANDS