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GENERAL
TITLE
REVEALING A MARINE NATURAL PRODUCT AS A NOVEL AGONIST FOR RETINOIC ACID RECEPTORS WITH A UNIQUE BINDING MODE AND ANTITUMOR ACTIVITY
DATE LAST MODIFIED
15 Nov 2017
RELEASE
3 Oct 2012
OBSOLETE
CLASSIFICATION
TRANSCRIPTION/TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 2 21 21
RESOLUTION RANGE HIGH
2.55
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1042/BJ20120726
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
A0QTG2 NR1B1, RARA ESCHERICHIA COLI HUMAN
RAR-ALPHA, NUCLEAR RECEPTOR SUBFAMILY 1 GROUP B ME ...
Q15788 -- -- HUMAN
NCOA-1, CLASS E BASIC HELIX-LOOP-HELIX PROTEIN 74, ...
Mutations
P10276 NR1B1, RARA ESCHERICHIA COLI HUMAN
RAR-ALPHA, NUCLEAR RECEPTOR SUBFAMILY 1 GROUP B ME ...
Mutations
Q15788 -- -- HUMAN
NCOA-1, CLASS E BASIC HELIX-LOOP-HELIX PROTEIN 74, ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402