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GENERAL
TITLE
CRYSTAL STRUCTURE OF DOT1L IN COMPLEX WITH EPZ003696
DATE LAST MODIFIED
9 Jan 2013
RELEASE
17 Oct 2012
OBSOLETE
CLASSIFICATION
TRANSFERASE/TRANSFERASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 65
RESOLUTION RANGE HIGH
2.8
RESOLUTION RANGE LOW
41.7
PUBMED ID
DOI
10.1111/CBDD.12050
PDBe
LIGANDS
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
P40302 | DOT1L, KIAA1814, KMT4 | ESCHERICHIA COLI | HUMAN | DOT1-LIKE PROTEIN, HISTONE H3-K79 METHYLTRANSFERAS ... |