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GENERAL
TITLE
N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH N-(1,1-DIOXO-1-THIAN-4-YL)- 5-METHYL-4-OXO-7-3-(TRIFLUOROMETHYL)PHENYL-4H,5H-THIENO-3,2-C- PYRIDINE-2-CARBOXIMIDAMIDE
DATE LAST MODIFIED
27 Sept 2017
RELEASE
22 Apr 2015
OBSOLETE
CLASSIFICATION
TRANSCRIPTION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
1.3
RESOLUTION RANGE LOW
39.32
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.5B00256
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P02554 -- ESCHERICHIA COLI HUMAN
PROTEIN HUNK1, HUMAN BRD4
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402