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GENERAL
TITLE
CRYSTAL STRUCTURE OF GSK-3BETA COMPLEXED WITH PF-04802367, A HIGHLY SELECTIVE BRAIN-PENETRANT KINASE INHIBITOR
DATE LAST MODIFIED
-
RELEASE
21 Sept 2016
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1 21 1
RESOLUTION RANGE HIGH
2.15
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1002/ANIE.201603797

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P0DTD1 GSK3B SPODOPTERA FRUGIPERDA HUMAN
GSK-3 BETA,SERINE/THREONINE-PROTEIN KINASE GSK3B
P49841 GSK3B SPODOPTERA FRUGIPERDA HUMAN
GSK-3 BETA,SERINE/THREONINE-PROTEIN KINASE GSK3B
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402