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3D Structure View

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GENERAL
TITLE
TRKA JM-KINASE WITH 1-(2-METHYL-4-PHENYL-PYRIMIDIN-5-YL)-3-[[2- (TRIFLUOROMETHYL)PHENYL]METHYL]UREA
DATE LAST MODIFIED
1 Feb 2017
RELEASE
28 Dec 2016
OBSOLETE
CLASSIFICATION
TRANSFERASE/TRANSFERASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 31 1 2
RESOLUTION RANGE HIGH
2.136
RESOLUTION RANGE LOW
44.3
PUBMED ID
DOI
10.1073/PNAS.1611577114
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
O50580 NTRK1, MTC, TRK, TRKA SPODOPTERA FRUGIPERDA HUMAN
NEUROTROPHIC TYROSINE KINASE RECEPTOR TYPE 1,TRK1- ...
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402