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3D Structure View

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GENERAL
TITLE
FACTOR VIIA IN COMPLEX WITH THE INHIBITOR (2R,15R)-2-[(1- AMINOISOQUINOLIN-6-YL)AMINO]-4,15,17-TRIMETHYL-7-[1-(1H-TETRAZOL-5- YL)CYCLOPROPYL]-13-OXA-4,11-DIAZATRICYCLO[14.2.2.1~6,10~]HENICOSA- 1(18),6(21),7,9,16,19-HEXAENE-3,12-DIONE
DATE LAST MODIFIED
12 Oct 2016
RELEASE
28 Sept 2016
OBSOLETE
CLASSIFICATION
HYDROLASE/HYDROLASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 41 21 2
RESOLUTION RANGE HIGH
1.73
RESOLUTION RANGE LOW
50
PUBMED ID
DOI
10.1016/J.BMCL.2016.08.088

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P08709 F7 CRICETINAE HUMAN
PROCONVERTIN,SERUM PROTHROMBIN CONVERSION ACCELERA ...
Mutations
P08709 F7 CRICETINAE HUMAN
PROCONVERTIN,SERUM PROTHROMBIN CONVERSION ACCELERA ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402