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GENERAL
TITLE
CRYSTAL STRUCTURE OF HUMAN PCAF BROMODOMAIN IN COMPLEX WITH COMPOUND-D (CPD-D), N-METHYL-2-(TETRAHYDRO-2H-PYRAN-4-YLOXY)BENZAMIDE
DATE LAST MODIFIED
11 Jan 2017
RELEASE
26 Oct 2016
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
H 3
RESOLUTION RANGE HIGH
2.05
RESOLUTION RANGE LOW
65.62
PUBMED ID
DOI
10.1021/ACSMEDCHEMLETT.6B00154
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q3HM40 KAT2B, PCAF ESCHERICHIA COLI HUMAN
HISTONE ACETYLTRANSFERASE PCAF,HISTONE ACETYLASE P ...
Q92831 KAT2B, PCAF ESCHERICHIA COLI HUMAN
HISTONE ACETYLTRANSFERASE PCAF,HISTONE ACETYLASE P ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402