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GENERAL
TITLE
THE CO-STRUCTURE OF (R)-4-(6-(1-(CYCLOPROPYLSULFONYL)CYCLOPROPYL)-2- (1H-INDOL-4-YL)PYRIMIDIN-4-YL)-3-METHYLMORPHOLINE AND A RATIONALLY DESIGNED PI3K-ALPHA MUTANT THAT MIMICS ATR
DATE LAST MODIFIED
-
RELEASE
14 Jun 2017
OBSOLETE
CLASSIFICATION
TRANSFERASE/SIGNALING PROTEIN/INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
2.5
RESOLUTION RANGE LOW
48.52
PUBMED ID
DOI
10.1016/J.JMB.2017.04.006
PDBe
LIGANDS