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6FEW

3D Structure View

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GENERAL
TITLE
DDR1, 2-[8-(1H-INDAZOLE-5-CARBONYL)-4-OXO-1-PHENYL-1,3,8- TRIAZASPIRO[4.5]DECAN-3-YL]-N-METHYLACETAMIDE, 1.440A, P1211, RFREE=24.1%
DATE LAST MODIFIED
27 Mar 2019
RELEASE
28 Nov 2018
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1 21 1
RESOLUTION RANGE HIGH
1.44
RESOLUTION RANGE LOW
43.42
PUBMED ID
DOI
10.1021/ACSCHEMBIO.8B00866
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q08345 DDR1, CAK, EDDR1, NEP, NTRK4, PTK3A, RTK6, TRKE SPODOPTERA FRUGIPERDA HUMAN
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1,CD167 ANTIG ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402