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GENERAL
TITLE
TARGETING MYELOID DIFFERENTIATION USING POTENT HUMAN DIHYDROOROTATE DEHYDROGENASE (HDHODH) INHIBITORS BASED ON 2-HYDROXYPYRAZOLO[1,5- A]PYRIDINE SCAFFOLD
DATE LAST MODIFIED
8 Aug 2018
RELEASE
11 Jul 2018
OBSOLETE
CLASSIFICATION
OXIDOREDUCTASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 32 2 1
RESOLUTION RANGE HIGH
1.58
RESOLUTION RANGE LOW
78.324
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.8B00373

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q02127 DHODH ESCHERICHIA COLI BL21(DE3) HUMAN
DHODEHASE,DIHYDROOROTATE OXIDASE
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402