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GENERAL
TITLE
RORCVAR2 (RORGT, 264-499) IN COMPLEX WITH COMPOUND 2 AT 2.3A: IDENTIFICATION OF N-ARYL IMIDAZOLES AS POTENT AND SELECTIVE RORGT INHIBITORS
DATE LAST MODIFIED
25 Dec 2019
RELEASE
27 Nov 2019
OBSOLETE
CLASSIFICATION
TRANSCRIPTION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 61 2 2
RESOLUTION RANGE HIGH
2.3
RESOLUTION RANGE LOW
19.64
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.9B01291
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
Q9UHD2 | RORC, NR1F3, RORG, RZRG | ESCHERICHIA COLI | HUMAN | NUCLEAR RECEPTOR RZR-GAMMA,NUCLEAR RECEPTOR SUBFAM ... |
NGL Viewer is used for the molecular visualization.
- AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
- AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402