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GENERAL
TITLE
RIP2 KINASE CATALYTIC DOMAIN COMPLEX WITH 2({4[(1,3BENZOTHIAZOL5YL) AMINO]6(2METHYLPROPANE2SULFONYL)QUINAZOLIN7YL}OXY)ETHAN1OL
DATE LAST MODIFIED
7 Aug 2019
RELEASE
17 Jul 2019
OBSOLETE
CLASSIFICATION
TRANSFERASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 32 2 1
RESOLUTION RANGE HIGH
2.62
RESOLUTION RANGE LOW
78.3
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.9B00575
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
O43353 RIPK2, CARDIAK, RICK, RIP2, UNQ277/PRO314/PRO34092 SPODOPTERA FRUGIPERDA HUMAN
CARD-CONTAINING INTERLEUKIN-1 BETA-CONVERTING ENZY ...
Mutations
O43353 RIPK2, CARDIAK, RICK, RIP2, UNQ277/PRO314/PRO34092 SPODOPTERA FRUGIPERDA HUMAN
CARD-CONTAINING INTERLEUKIN-1 BETA-CONVERTING ENZY ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402