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GENERAL
TITLE
HIF PROLYL HYDROXYLASE 2 (PHD2/ EGLN1) IN COMPLEX WITH 4-HYDROXY-N-(4- PHENOXYBENZYL)-2-(1H-PYRAZOL-1-YL)PYRIMIDINE-5-CARBOXAMIDE
DATE LAST MODIFIED
19 Feb 2020
RELEASE
4 Dec 2019
OBSOLETE
CLASSIFICATION
OXIDOREDUCTASE
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 2 21
RESOLUTION RANGE HIGH
2.426
RESOLUTION RANGE LOW
83.92
PUBMED ID
DOI
10.1002/CMDC.201900557
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q9GZT9 EGLN1, C1ORF12, PNAS-118, PNAS-137 ESCHERICHIA COLI BL21(DE3) HUMAN
HYPOXIA-INDUCIBLE FACTOR PROLYL HYDROXYLASE 2,HPH- ...
Mutations
Q9GZT9 EGLN1, C1ORF12, PNAS-118, PNAS-137 ESCHERICHIA COLI BL21(DE3) HUMAN
HYPOXIA-INDUCIBLE FACTOR PROLYL HYDROXYLASE 2,HPH- ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402