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GENERAL
TITLE
DYRK1A BOUND TO A HARMINE DERIVATIVE
DATE LAST MODIFIED
8 Apr 2020
RELEASE
12 Feb 2020
OBSOLETE
CLASSIFICATION
TRANSFERASE/TRANSFERASE INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 1 2 1
RESOLUTION RANGE HIGH
2.95
RESOLUTION RANGE LOW
125.9
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.9B01379
PDBe
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Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P21853 DYRK1A, DYRK, MNB, MNBH ESCHERICHIA COLI BL21 HUMAN
DUAL SPECIFICITY YAK1-RELATED KINASE,HP86,PROTEIN ...
Q13627 DYRK1A, DYRK, MNB, MNBH ESCHERICHIA COLI BL21 HUMAN
DUAL SPECIFICITY YAK1-RELATED KINASE,HP86,PROTEIN ...
Mutations
P21852 DYRK1A, DYRK, MNB, MNBH ESCHERICHIA COLI BL21 HUMAN
DUAL SPECIFICITY YAK1-RELATED KINASE,HP86,PROTEIN ...
Q13627 DYRK1A, DYRK, MNB, MNBH ESCHERICHIA COLI BL21 HUMAN
DUAL SPECIFICITY YAK1-RELATED KINASE,HP86,PROTEIN ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402