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GENERAL
TITLE
ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN Y537S MUTANT IN COMPLEX WITH A METHYLATED LASOFOXIFENE DERIVATIVE THAT POSSESSES SELECTIVE ESTROGEN RECEPTOR DEGRADER ACTIVITIES
DATE LAST MODIFIED
-
RELEASE
1 Apr 2020
OBSOLETE
CLASSIFICATION
TRANSCRIPTION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 1
RESOLUTION RANGE HIGH
2.59
RESOLUTION RANGE LOW
50
PUBMED ID
-
DOI
--
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P03372 ESR1, ESR, NR3A1 ESCHERICHIA COLI HUMAN
ER,ER-ALPHA,ESTRADIOL RECEPTOR,NUCLEAR RECEPTOR SU ...
P03372 ESR1, ESR, NR3A1 ESCHERICHIA COLI HUMAN
ER,ER-ALPHA,ESTRADIOL RECEPTOR,NUCLEAR RECEPTOR SU ...
P03372 ESR1, ESR, NR3A1 ESCHERICHIA COLI HUMAN
ER,ER-ALPHA,ESTRADIOL RECEPTOR,NUCLEAR RECEPTOR SU ...
P03372 ESR1, ESR, NR3A1 ESCHERICHIA COLI HUMAN
ER,ER-ALPHA,ESTRADIOL RECEPTOR,NUCLEAR RECEPTOR SU ...
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402