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GENERAL
TITLE
KEAP1 KELCH DOMAIN BOUND TO A SMALL MOLECULE INHIBITOR OF THE KEAP1- NRF2 PROTEIN-PROTEIN INTERACTION
DATE LAST MODIFIED
5 May 2021
RELEASE
14 Apr 2021
OBSOLETE
CLASSIFICATION
PEPTIDE BINDING PROTEIN
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 61
RESOLUTION RANGE HIGH
1.75
RESOLUTION RANGE LOW
44.75
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.0C02094
PDBe
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LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
Q8RQE9 KEAP1, INRF2, KIAA0132 ESCHERICHIA COLI 'BL21-GOLD(DE3)PLYSS AG' MOUSE
CYTOSOLIC INHIBITOR OF NRF2,INRF2
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402